PHENOXYMETHYL DERIVATIVES Russian patent published in 2021 - IPC C07D403/12 C07D231/12 C07D231/56 C07D401/12 C07D237/14 C07D407/04 C07D407/12 C07D409/12 C07D413/12 C07D417/12 C07D249/12 C07D471/04 C07D487/04 C07F7/08 A61K31/4162 A61K31/4192 A61K31/4196 A61K31/415 A61K31/4245 A61K31/50 A61K31/695 A61P27/02 

Abstract RU 2746481 C1

FIELD: pharmacology.

SUBSTANCE: present invention relates to a compound of Formula (I) or a pharmaceutically acceptable salt thereof, as well as to a specific phenoxymethyl derivative or a pharmaceutically acceptable salt thereof having the ability to inhibit ATC, to a pharmaceutical composition containing them, to their use and to a method for inhibiting ATC

In Formula I, W is selected from ring systems A, B, C, D and E:

wherein RA, RB, RC, RC1, RD1, RD4, A1-A6 are such as defined in the claim.

EFFECT: ATC inhibiting.

38 cl, 30 tbl, 221 ex

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Authors

Khert Zherom

Khuntsiker Daniel

Kyune Kholger

Lyubbers Tomas

Martin Rajner E.

Mattej Patritsio

Najdkhart Verner

Rikhter Khans

Rudolf Markus

Pinar Emmanyuel

Dates

2021-04-14Published

2016-09-01Filed