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RU

(11)

2 748 838

(13)

C2

(51)

IPC

C07C259/06(2006-01-01)

A61K31/201(2006-01-01)

A61P35/00(2006-01-01)

C07C229/34(2006-01-01)

C07C235/42(2006-01-01)

C07C251/40(2006-01-01)

C07C251/48(2006-01-01)

C07C251/60(2006-01-01)

C07C271/20(2006-01-01)

C07C271/22(2006-01-01)

C07C279/14(2006-01-01)

C07C279/24(2006-01-01)

C07C323/41(2006-01-01)

C07C403/20(2006-01-01)

C07C59/72(2006-01-01)

C07C59/74(2006-01-01)

C07C59/90(2006-01-01)

C07D215/12(2006-01-01)

C07D215/28(2006-01-01)

(21) (22)

Application

2019112675, 2017-09-28

(24)

Start date

2017-09-28

(22)

Actual filing date

2017-09-28

(45)

Published

2021-05-31

(72)

Inventor

Pisano, ClaudioDallavalle, SabrinaCincinelli, RaffaellaMerlini, Lucio

(73)

Holder

Biogem S.C. A R.L.

RETINOID DERIVATIVES WITH ANTITUMOR ACTIVITY Russian patent published in 2021 - IPC C07C259/06 A61K31/201 A61P35/00 C07C229/34 C07C235/42 C07C251/40 C07C251/48 C07C251/60 C07C271/20 C07C271/22 C07C279/14 C07C279/24 C07C323/41 C07C403/20 C07C59/72 C07C59/74 C07C59/90 C07D215/12 C07D215/28 

Abstract RU 2748838 C2

FIELD: biochemistry.

SUBSTANCE: present invention relates to compounds of Formula (I) and to pharmaceutical compositions containing them:

wherein the values of substituents are indicated in the claims. Such compounds for use in the treatment of cancer and other diseases associated with altered angiogenesis, such as pathologies related to arthritis, diabetic retinopathy, psoriasis and chronic inflammatory disease, are also included in the scope of the present invention.

EFFECT: invention can be used in treatment of cancer and other diseases associated with altered angiogenesis, such as pathologies related to arthritis, diabetic retinopathy, psoriasis and chronic inflammatory disease.

10 cl, 11 tbl, 1 dwg, 23 ex

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RU 2 748 838 C2

Authors

Pisano, Claudio

Dallavalle, Sabrina

Cincinelli, Raffaella

Merlini, Lucio

Dates

2021-05-31—Published

2017-09-28—Filed

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