AMORPHOUS DERIVATIVE OF PYRROLIDINE AS PPAR AGONIST AND METHOD FOR PRODUCTION THEREOF Russian patent published in 2021 - IPC C07D207/06 A61K31/4025 A61P1/16 

Abstract RU 2749056 C1

FIELD: chemistry.

SUBSTANCE: invention relates to an amorphous form of the compound represented by the formula (I) wherein the powder X-ray diffractogram of the amorphous form does not have any sharp diffraction peak and has a wide reclined diffraction peak at an angle of 2θ between 10° and 25°, as well as to a method of production thereof.

EFFECT: new amorphous form of the compound represented by the formula (I) is produced which can be used as a PPAR agonist, wherein the amorphous form is characterized by significant stability.

7 cl, 3 dwg, 5 tbl, 3 ex

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RU 2 749 056 C1

Authors

Yujan, Chzhilyan

Tszyan, Chzhigan

Khe, Khajin

Chzhan, Syao

Syuj, Tsziven

Chzho, Vejsyan

Li, Tszyan

Chen, Shukhoj

Dates

2021-06-03Published

2018-12-20Filed