NOVEL AGONIST OF β-RECEPTOR OF THYROID HORMONES Russian patent published in 2025 - IPC C07D239/34 C07D239/02 C07D403/12 A61K31/505 A61K31/506 A61P3/04 A61P3/06 A61P5/14 

Abstract RU 2839610 C1

FIELD: chemistry.

SUBSTANCE: invention relates to novel agonists β-receptor of thyroid hormones of formula (I) and their use for preventing or treating diseases associated with action of an agonist β-receptor, wherein said disease includes, for example, obesity, hyperlipidemia, hypercholesterolemia, diabetes, liver disease, particularly fatty hepatosis, NASH, NAFLD, cardiovascular diseases, in particular atherosclerosis, thyroid diseases, in particular hypothyroidism or thyroid cancer. $$$ Formula I.

EFFECT: compounds have better activity, selectivity or safety.

16 cl, 2 dwg, 10 tbl, 52 ex

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RU 2 839 610 C1

Authors

Yuj, Yungo

Van, Itsyan

Ke, Tszunkhun

Dates

2025-05-06Published

2021-06-02Filed