FIELD: chemistry.
SUBSTANCE: invention relates to novel agonists β-receptor of thyroid hormones of formula (I) and their use for preventing or treating diseases associated with action of an agonist β-receptor, wherein said disease includes, for example, obesity, hyperlipidemia, hypercholesterolemia, diabetes, liver disease, particularly fatty hepatosis, NASH, NAFLD, cardiovascular diseases, in particular atherosclerosis, thyroid diseases, in particular hypothyroidism or thyroid cancer. $$$ Formula I.
EFFECT: compounds have better activity, selectivity or safety.
16 cl, 2 dwg, 10 tbl, 52 ex
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Authors
Dates
2025-05-06—Published
2021-06-02—Filed