FIELD: pharmaceuticals.
SUBSTANCE: invention relates to a pharmaceutical composition based on 6-amino-9-[(3R)-1-(2-butinoyl)-3-pyrrolidinyl]-7-(4-phenoxyphenyl)-7,9-dihydro-8H-purine-8-one hydrochloride, which has the activity of a selective Btk inhibitor, useful for the prevention and/or treatment of Btk-related diseases. The invention also relates to the use of 6-amino-9-[(3R)-1-(2-butinoyl)-3-pyrrolidinyl]-7-(4-phenoxyphenyl)-7,9-dihydro-8H-purine-8-one hydrochloride.
EFFECT: pharmaceutical composition based on a Btk inhibitor has been obtained that is useful for the treatment of non-Hodgkin's lymphoma, autoimmune disease, and other Btk-related diseases.
6 cl, 4 dwg, 6 tbl, 15 ex
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Authors
Dates
2021-06-29—Published
2012-11-28—Filed