ANTIVIRAL ALIPHATIC ESTER PRODRUGS OF TENOFOVIR Russian patent published in 2021 - IPC C07D473/34 C07F9/6561 A61K31/52 A61K31/675 A61K45/06 A61P31/18 

Abstract RU 2759902 C2

FIELD: medicine.

SUBSTANCE: present invention relates to aliphatic ester prodrugs of tenofovir, namely to a group of compounds indicated in the claim of the invention that have antiviral activity relatively to HIV-1. A pharmaceutical composition for inhibiting reverse HIV transcriptase is also proposed.

EFFECT: obtaining new compounds suitable for use in the prevention or treatment of HIV infection.

7 cl, 4 tbl, 17 ex

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RU 2 759 902 C2

Authors

Raheem, Izzat

Paparin, Jean-Laurent

Rahali, Houcine

Da Costa, Daniel

Dukhan, David

Dates

2021-11-18Published

2017-12-20Filed