FIELD: medicine; pharmaceuticals.
SUBSTANCE: invention relates to a compound of formula I or a pharmaceutically acceptable salt thereof, useful in pharmaceutics and medicine:
,
where: R1 is -H, -C(O)R3 or , R2 is -H or -C(O)R4; each of R3 and R4 is independently selected from -(C1-C3alkylene)m-(C6-C10aryl), where aryl is unsubstituted or substituted with substituent R5; m is integer 1; R5 is -C1-C6 alkyl.
EFFECT: what is presented is a novel compound, a based pharmaceutical composition and a method thereof, which are effective for treating and preventing HIV infection.
14 cl, 6 tbl, 4 ex
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Authors
Dates
2020-05-13—Published
2016-09-19—Filed