FUCOSIDASE INHIBITORS Russian patent published in 2022 - IPC C07D211/46 C07D211/74 A61K31/445 A61K45/06 A61K9/19 A61P35/00 

Abstract RU 2765202 C2

FIELD: medicine.

SUBSTANCE: invention relates to a compound of the formula I having properties of fucosidase enzyme inhibitors and its use for the treatment of tumor or cancer disease, which is liver cancer. In the general formula I, X1, X2 and X3 are OH; R is C1-3alkyl; R1 is H; R2 is selected from a group consisting of -NRbC(O)Ra, and -C(O)NRbRa; Ra is ; and Rb is H.

EFFECT: obtaining fucosidase inhibitors.

(I)

8 cl, 3 dwg, 9 tbl, 10 ex

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RU 2 765 202 C2

Authors

Zankel, Todd, C.

Isbell, Sara, Louise

Ko, Amanda, Anne

Dates

2022-01-26Published

2016-07-29Filed