Show metadata Hide metadata

(19)

(11)

2 766 543

(13)

(51)

IPC

C07D245/04(2006-01-01)

C07K5/02(2006-01-01)

C07K5/08(2006-01-01)

C07K5/10(2006-01-01)

C07K7/00(2006-01-01)

A61K31/395(2006-01-01)

A61K31/407(2006-01-01)

A61K31/4196(2006-01-01)

A61K31/496(2006-01-01)

A61K38/06(2006-01-01)

A61K38/07(2006-01-01)

A61K38/08(2006-01-01)

A61P31/04(2006-01-01)

(21) (22)

Application

2018122505, 2016-11-21

(24)

Start date

2016-11-21

(22)

Actual filing date

2016-11-21

(45)

Published

2022-03-15

(72)

Inventor

Chen, YunshenSmit, Peter EndryuRoberts, Taker KarranKhiguchi, Robert I.Paraselli, PrasunaKeler, Majkl F.T.Shvarts, Dzhejkob BredliKrouford, Dzhejms DzhonLyu, Kuong Ts.Khenen, Emili Dzh.Khu, KhuajongYuj,Chzhioyun

(73)

Holder

Arkyuiks Farmasyutikels, Ink.Dzhenetek, Ink.

MACROCYCLIC ANTIBIOTICS OF WIDE RANGE OF ACTIONS Russian patent published in 2022 - IPC C07D245/04 C07K5/02 C07K5/08 C07K5/10 C07K7/00 A61K31/395 A61K31/407 A61K31/4196 A61K31/496 A61K38/06 A61K38/07 A61K38/08 A61P31/04

Abstract RU 2766543 C2

FIELD: medicine.

SUBSTANCE: invention relates to compounds selected from a group consisting of compounds 101, 102, 103, 104, etc. that relate to macrocyclic antibiotics of a wide range of actions and that can be used for the treatment of various bacterial infections. The invention also relates to a pharmaceutical composition and a method for the treatment of a bacterial infection using the specified compounds.

EFFECT: obtaining compounds for the treatment of bacterial infections.

, ,

4 cl, 1 dwg, 2 tbl, 432 ex

Similar patents RU2766543C2

Title	Year	Author	Number
MACROCYCLIC WIDE-RANGE ANTIBIOTICS	2018	Smith, Peter, Andrew Roberts, Tucker, Curran Higuchi, Robert, I. Paraselli, Prasuna Koehler, Michael, F., T. Schwarz, Jacob, Bradley Crawford, James, John Ly, Cuong Q. Hanan, Emily, J. Hu, Huiyong Chen, Yongsheng Yu, Zhiyong Winship, Paul Colin Michael Mccleod, Calum Blench, Toby	RU2779477C2
MACROCYCLIC ANTIBIOTICS OF WIDE SPECTRUM OF ACTION	2016	Chen Yunshen Smit Peter Endryu Roberts Taker Karran Khiguchi Robert I. Paraselli Prasuna Keler Majkl F.T. Shvarts Dzhejkob Bredli Krouford Dzhejms Dzhon Lyu Kuong Ts. Khu Khuajong Yuj Chzhioyun	RU2761476C2
BICYCLIC AGONISTS OF THE INTERFERON GENE STIMULATOR STING	2020	Petrassi, Khenk Majkl Dzhejms Yuj, Chenian Van, Tsze Chatterdzhi, Arnab K. Shults, Piter Dzh. Dzhonson, Kristen Chu, Alan Chin, Emili Lejrson, Lyuk L.	RU2800072C1
NEW ACTIVATORS OF SOLUBLE GUANYLATE CYCLASE AND PHOSPHODIESTERASE INHIBITORS WITH DUAL ACTION MECHANISM AND THEIR APPLICATION	2018	Naef, Reto Tenor, German	RU2758373C2
CEREBLON LIGANDS AND BIFUNCTIONAL COMPOUNDS CONTAINING THEM	2018	Crew, Andrew, P. Berlin, Michael Dong, Hanqing Hornberger, Keith, R. Qian, Yimin Snyder, Lawrence, B. Wang, Jing Zimmermann, Kurt	RU2795146C2
INHIBITORS OF CDK	2011	Tavares Fransis Kh. Strum Dzhej S.	RU2621674C2
PYRAZOLE-BASED MAGL INHIBITORS	2018	Grajs, Sheril A. Viner, Dzhon Dzh.M. Veber, Oliviya D. Dunkan Katarina K.	RU2789157C2
ANALOGUES OF 4H-PYRAZOLO[1,5-A]BENZIMIDAZOLE COMPOUNDS AS PARP INHIBITORS	2015	Van Syuekhaj Din Chzhaochzhun Syuj Yun Chen Shukhuej Li Le Li Gan Tu Zhunkhua Van Tsajlin Yue Yan Chzhan Chzhibo Chen Khajlyan Sun Ventsze Khuan Lu	RU2672722C2
MEK INHIBITORS AND THEIR THERAPEUTIC USE	2021	Kholl, Brett Mettyu Dekorte, Bart Liven King, Piter Dzhon Linders, Ruben Vegert, Anita Fouler, Kevin Kolitts, Sara Dudman, Robin Polakker, Yarno Folmer, Rutger Khenk Adrian	RU2812929C1
OESTROGEN RECEPTOR MODULATING COMPOUNDS	2019	Miller, Kris	RU2826635C2

RU 2 766 543 C2

Authors

Chen, Yunshen

Smit, Peter Endryu

Roberts, Taker Karran

Khiguchi, Robert I.

Paraselli, Prasuna

Keler, Majkl F.T.

Shvarts, Dzhejkob Bredli

Krouford, Dzhejms Dzhon

Lyu, Kuong Ts.

Khenen, Emili Dzh.

Khu, Khuajong

Yuj,Chzhioyun

Dates

2022-03-15—Published

2016-11-21—Filed