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(19)

(11)

2 766 543

(13)

(51)

IPC

C07D245/04(2006-01-01)

C07K5/02(2006-01-01)

C07K5/08(2006-01-01)

C07K5/10(2006-01-01)

C07K7/00(2006-01-01)

A61K31/395(2006-01-01)

A61K31/407(2006-01-01)

A61K31/4196(2006-01-01)

A61K31/496(2006-01-01)

A61K38/06(2006-01-01)

A61K38/07(2006-01-01)

A61K38/08(2006-01-01)

A61P31/04(2006-01-01)

(21) (22)

Application

2018122505, 2016-11-21

(24)

Start date

2016-11-21

(22)

Actual filing date

2016-11-21

(45)

Published

2022-03-15

(72)

Inventor

Chen, YunshenSmit, Peter EndryuRoberts, Taker KarranKhiguchi, Robert I.Paraselli, PrasunaKeler, Majkl F.T.Shvarts, Dzhejkob BredliKrouford, Dzhejms DzhonLyu, Kuong Ts.Khenen, Emili Dzh.Khu, KhuajongYuj,Chzhioyun

(73)

Holder

Arkyuiks Farmasyutikels, Ink.Dzhenetek, Ink.

MACROCYCLIC ANTIBIOTICS OF WIDE RANGE OF ACTIONS Russian patent published in 2022 - IPC C07D245/04 C07K5/02 C07K5/08 C07K5/10 C07K7/00 A61K31/395 A61K31/407 A61K31/4196 A61K31/496 A61K38/06 A61K38/07 A61K38/08 A61P31/04

Abstract RU 2766543 C2

FIELD: medicine.

SUBSTANCE: invention relates to compounds selected from a group consisting of compounds 101, 102, 103, 104, etc. that relate to macrocyclic antibiotics of a wide range of actions and that can be used for the treatment of various bacterial infections. The invention also relates to a pharmaceutical composition and a method for the treatment of a bacterial infection using the specified compounds.

EFFECT: obtaining compounds for the treatment of bacterial infections.

, ,

4 cl, 1 dwg, 2 tbl, 432 ex

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RU 2 766 543 C2

Authors

Chen, Yunshen

Smit, Peter Endryu

Roberts, Taker Karran

Khiguchi, Robert I.

Paraselli, Prasuna

Keler, Majkl F.T.

Shvarts, Dzhejkob Bredli

Krouford, Dzhejms Dzhon

Lyu, Kuong Ts.

Khenen, Emili Dzh.

Khu, Khuajong

Yuj,Chzhioyun

Dates

2022-03-15—Published

2016-11-21—Filed