FIELD: pharmaceuticals.
SUBSTANCE: invention relates to a compound by the general formula (I), exhibiting an analgesic or anti-inflammatory effect. In the formula (I), both R are the same and constitute an ethyl group or a residue of an ester of (L)-malic acid. The invention also relates to an application of compounds by the general formula (I), wherein both R are the same and constitute hydrogen, an ethyl group, or a residue of an ester of (L)-malic acid, as an analgesic or anti-inflammatory agent, as inhibitors of ASIC1a and ASIC3 ion channels, or as a medicinal product for preventing or treating pain and inflammation. (I).
EFFECT: creation of a compound with an analgesic or anti-inflammatory effect.
7 cl, 15 dwg, 19 ex
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Authors
Dates
2022-05-16—Published
2020-10-22—Filed