FIELD: pharmaceutical industry.
SUBSTANCE: invention relates to new anxiolytic agents, namely N-substituted 4-(1-hydroxy-1-methyl-2-aminoethyl)benzoic acids of the general formula (1), their pharmaceutically acceptable salts. The invention also relates to a method for obtaining compounds, consisting in the implementation of three stages.
EFFECT: compounds of the general formula (1) having a pronounced anxiolytic effect with low toxicity with no sedative effect and excitatory effect on the central nervous system.
where R=H, -CnH2n+1 (n=1-6),
(n=1-4),
2 cl, 9 ex, 4 tbl
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