BENZIMIDAZOLE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS Russian patent published in 2022 - IPC C07D403/12 C07D403/14 C07D405/14 C07D413/14 C07D401/12 C07D487/10 C07D498/10 C07D235/30 C07D235/32 A61K31/4184 A61P31/00 A61P35/00 

Abstract RU 2781429 C2

FIELD: medicine.

SUBSTANCE: invention relates to benzimidazole derivatives, a pharmaceutical preparation containing the specified derivatives, which is intended for the treatment and/or prevention of physiological and/or pathophysiological conditions mediated by activity of an adenosine receptor A2A or adenosine receptors A2A and A2B, for example, such as hyperproliferative or infectious diseases and disorders.

EFFECT: obtaining benzimidazole derivatives for the treatment of diseases.

11 cl, 7 tbl, 9 ex

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RU 2 781 429 C2

Authors

Tanzer Eva-Maria

Schiemann Kai

Klein Markus

Dates

2022-10-11Published

2018-08-20Filed