THIAZOLOPYRIDINE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS Russian patent published in 2023 - IPC C07D513/04 C07D519/00 A61K31/437 A61K31/4365 A61P35/00 

Abstract RU 2810114 C2

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to specific thiazolopyridine derivatives specified in paragraph 1 of the formula, as well as to a pharmaceutical preparation and a medicinal product based on these derivatives for inhibiting adenosine receptors A2A and/or A2B.

EFFECT: new compounds and medicinal products based on them have been obtained, the said compounds and medicinal products can be used in medicine for the treatment or prevention of hyperproliferative or infectious diseases and disorders.

10 cl, 10 tbl, 10 ex

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RU 2 810 114 C2

Authors

Tanzer Eva-Maria

Schiemann Kai

Crespo Alejandro

Dates

2023-12-21Published

2020-01-21Filed