FIELD: pharmaceuticals.
SUBSTANCE: invention relates to specific thiazolopyridine derivatives specified in paragraph 1 of the formula, as well as to a pharmaceutical preparation and a medicinal product based on these derivatives for inhibiting adenosine receptors A2A and/or A2B.
EFFECT: new compounds and medicinal products based on them have been obtained, the said compounds and medicinal products can be used in medicine for the treatment or prevention of hyperproliferative or infectious diseases and disorders.
10 cl, 10 tbl, 10 ex
Title |
Year |
Author |
Number |
THIAZOLOPYRIDINE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS |
2018 |
- Tanzer Eva-Maria
- Schiemann Kai
- Klein Markus
|
RU2790011C2 |
QUINOXALINE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS |
2018 |
- Tanzer Eva-Maria
- Schiemann Kai
- Klein Markus
|
RU2791168C1 |
BENZIMIDAZOLE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS |
2018 |
- Tanzer Eva-Maria
- Schiemann Kai
- Klein Markus
|
RU2781429C2 |
PYRAZOLOPYRIMIDINE COMPOUNDS AS ADENOSINE RECEPTOR ANTAGONISTS |
2019 |
- Bell, Andrew Simon
- Schreyer, Adrian Michael
- Versluys, Stephanie
|
RU2806758C2 |
SUBSTITUTED PHENOXYACETIC ACIDS, THEIR ESTERS AND AMIDES CONTAINING 2,6-DIOXO-2,3,6,7-TETRAHYDRO-1H-PYRIN-8-YL FRAGMENTS - A ADENOSINE RECEPTOR ANTAGONISTS AND USE THEREOF |
2011 |
- Ivashchenko Aleksandr Vasil'Evich
- Mit'Kin Oleg Dmitrievich
- Kadieva Madina Georgievna
- Okun' Il'Ja Matusovich
|
RU2477726C1 |
SUBSTITUTED 1,3-DIETHYL-8-VINYL-7-METHYL-3,7-DIHYDROPURINE-2,6-DIONES - ANTAGONISTS OF ADENOSINE A RECEPTOR AND USE THEREOF |
2012 |
- Ivashchenko Aleksandr Vasil'Evich
|
RU2480469C1 |
DERIVATIVES OF BENZOTHIAZOLE AND MEDICAMENT BASED ON THEREOF |
2002 |
- Flor Aleksander
- Jakob-Retne Roland
- Norkross David Rozhe
- Rimer Klaus
|
RU2293083C2 |
DERIVATIVES OF 8-METHOXY-[1,2,4]TRIAZOLO[1,5-a]PYRIDINE AND PHARMACEUTICAL PREPARATION BASED ON THEREOF |
2002 |
- Nettekofen Mattias Genrikh
- Pjull'Mann Bernd
|
RU2297416C2 |
2-AMINOBENZOTHIAZOLYLUREAS AS ADENOSINE MODULATORS |
2002 |
- Flor Aleksander
- Jakob-Retne Roland
- Norkross Rozhe David
- Rimer Klaus
|
RU2311905C2 |
BENZOTHIOPHENES AS MODULATORS OF ADENOSINE RECEPTORS |
2002 |
- Alanin Aleksander
- Flor Aleksander
|
RU2299882C2 |