QUINOXALINE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS Russian patent published in 2023 - IPC C07D241/44 C07D403/04 C07D403/12 C07D405/04 C07D413/14 C07D417/14 C07D471/04 C07D495/10 A61K31/498 A61K45/06 A61P31/00 A61P35/00 

Abstract RU 2791168 C1

FIELD: pharmaceutics.

SUBSTANCE: invention relates to quinoxaline derivatives, namely to a group of individual compounds, such as those specified in the claims of the invention. A pharmaceutical preparation and a method for its preparation, a medicinal product are also proposed.

EFFECT: proposed compounds are highly effective inhibitors of adenosine receptor A2A or adenosine receptors A2A and A2B and can be used for the treatment and/or prevention of physiological and/or pathophysiological conditions selected from a group consisting of hyperproliferative and infectious diseases and disorders mediated by the activity of an inhibitor of adenosine receptors A2A and/or A2B.

10 cl, 7 tbl, 9 ex

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RU 2 791 168 C1

Authors

Tanzer Eva-Maria

Schiemann Kai

Klein Markus

Dates

2023-03-03Published

2018-08-20Filed