THIAZOLOPYRIDINE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS Russian patent published in 2023 - IPC C07D513/04 A61P31/00 A61P35/00 

Abstract RU 2790011 C2

FIELD: biotechnology.

SUBSTANCE: invention relates to thiazolopyridine derivatives of the general formula I, as well as to methods for their production and the use as A2A and/or A2B adenosine receptor inhibitor.

EFFECT: new compounds are obtained, which can be used for the treatment and/or prevention of hyperproliferative or infectious diseases mediated with inhibition of A2A and/or A2B adenosine receptor.

14 cl, 7 tbl, 9 ex

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RU 2 790 011 C2

Authors

Tanzer Eva-Maria

Schiemann Kai

Klein Markus

Dates

2023-02-14Published

2018-07-02Filed