6-OXO-3-PHENYL-2-(PHENYLAMINO)-3,4,5,6-TETRAHYDROPYRIMIDINE-4-CARBOXYLIC ACID AND METHOD FOR ITS PRODUCTION Russian patent published in 2022 - IPC C07D239/22 A61K31/513 A61P29/00 

Abstract RU 2785763 C1

FIELD: organic chemistry.

SUBSTANCE: invention relates to the field of organic chemistry, namely to 6-oxo-3-phenyl-2-(phenylamino)-3,4,5,6-tetrahydropyrimidine-4-carboxylic acid of the formula I and to a method for its preparation. The method is carried out by the interaction of diphenylguanidine with maleic anhydride in a molar ratio of 1:1.17, respectively, in a methylene chloride medium for 15 minutes.

EFFECT: obtaining a new chemical compound that has analgesic and anti-inflammatory activity.

2 cl, 1 dwg, 4 tbl, 3 ex

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RU 2 785 763 C1

Authors

Trukhanova Yuliya Aleksandrovna

Kolesnik Denis Andreevich

Yuskovets Valerij Nikolaevich

Kuvaeva Elena Vladimirovna

Ksenofontova Galina Vladimirovna

Semakova Tamara Leonidovna

Yakovlev Igor Pavlovich

Dates

2022-12-12Published

2022-04-20Filed