FIELD: medicine.
SUBSTANCE: group of inventions refers to a water-soluble agent based on polygalacturonate, which has selective cytotoxic activity against A549 lung carcinoma, MCF-7 breast adenocarcinoma and M-HeLa cervical carcinoma, which is potassium cobalt polygalacturonate (PCCo) or its composition with sodium-cobalt-polygalacturonate (PNaCo) in a mass ratio of 1-2:1-2, and also refers to a water-soluble polygalacturonate-based agent with selective cytotoxic activity against A549 lung carcinoma, MCF-7 breast adenocarcinoma and cervical carcinoma M-HeLa, which is a composition containing sodium-cobalt-polygalacturonate (PNaCo) in a mass ratio of 3:1 and a metal complex of pectin biopolymer sodium-metal-polygalacturonate, respectively, where the biogenic metal is zinc, manganese, chromium or magnesium (PGNaZn, PGNaMn, PGNaCr, PGNaMg).
EFFECT: obtaining antitumor agents based on macro- and microelement-containing polygalacturonates.
2 cl, 1 dwg, 3 tbl
| Title | Year | Author | Number | 
|---|---|---|---|
| SODIUM COBALT POLYGALACTURONATE WITH ANTITUMOR ACTIVITY | 2023 | 
 | RU2794885C1 | 
| NEW STERICALLY HINDERED PHENOLS CONTAINING BENZOFUROXAN FRAGMENTS WITH ANTITUMOR ACTIVITY | 2022 | 
 | RU2796810C1 | 
| BROMINE-CONTAINING STERICALLY HINDERED PHENOLS WITH ANTICANCER ACTIVITY | 2023 | 
 | RU2822270C1 | 
| LOW-TOXICITY AMINOPHOSPHONIUM SALTS HAVING ANTICANCER ACTIVITY, AND METHOD FOR PREPARING THEM | 2024 | 
 | RU2836726C1 | 
| CONJUGATE OF ANTITUMOUR DRUGS WITH RECOMBINANT ALPHA-FETOPROTEIN AND ITS FUNCTIONAL FRAGMENTS AND METHOD OF THEIR PRODUCING | 2016 | 
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| MIXED-LIGAND COMPLEXES OF COPPER (II) WITH 1H-TETRAZOLE-5-ACETIC ACID AND OLIGOPYRIDINE DERIVATIVES, EXHIBITING CYTOTOXIC ACTIVITY | 2023 | 
 | RU2818953C1 | 
| AGENT BASED ON ARGLABIN DERIVATIVE, HAVING SELECTIVE CYTOTOXIC ACTION | 2023 | 
 | RU2814259C1 | 
| THE USE OF CARRIMYCIN AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS FOR THE PRODUCTION OF MEDICINES FOR TREATMENT AND / OR TUMOR PREVENTION | 2018 | 
 | RU2746047C1 | 
| METHODS AND COMPOSITIONS FOR TREATING CANCER | 2009 | 
 | RU2508116C2 | 
| PINANE C,N-PALLADACYCLES CONTAINING L-AMINO ACIDS AND THEIR USE AS ANTITUMOR AGENTS | 2022 | 
 | RU2799205C1 | 
Authors
Dates
2023-03-22—Published
2022-06-23—Filed