PYRIMIDOIMIDAZOLE COMPOUNDS USED AS DNA-RK INHIBITORS Russian patent published in 2023 - IPC A61K31/522 A61P35/00 C07D473/18 C07D487/04 C07D519/00 

Abstract RU 2796163 C1

FIELD: medicine.

SUBSTANCE: group of inventions exhibits a therapeutic effect on solid and hematological tumors. Derivatives of the compound of formula (IV) are provided. In another embodiment, the use of the said compounds in the manufacture of a DNA-RK inhibitor is provided.

EFFECT: group of inventions provides new derivatives of compounds of formula (IV) having inhibitory activity against DNA-RK.

14 cl, 1 dwg, 8 tbl, 31 ex

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RU 2 796 163 C1

Authors

Chen, Kevin X

Xia, Shanghua

Chen, Zhaoguo

Guo, Zuhao

Yu, Yanxin

Zhou, Kai

Hu, Boyu

Zhang, Li

Jiang, Fen

Wang, Jingjing

Hu, Guoping

Li, Jian

Chen, Shuhui

Dates

2023-05-17Published

2020-11-25Filed