THIAZOLACTAM COMPOUNDS AS ERK INHIBITORS AND THEIR APPLICATIONS Russian patent published in 2023 - IPC C07D513/04 A61K31/506 A61P35/00 

Abstract RU 2805569 C1

FIELD: thiazolactam compounds.

SUBSTANCE: invention is related to thiazolactam compounds of formula (III), where the values of R1-R5, n, m are defined in the claims.

EFFECT: used in preparation of drugs for treatment of diseases associated with ERK.

16 cl, 2 dwg, 6 tbl, 13 ex

Similar patents RU2805569C1

Title Year Author Number
SPIRO COMPOUNDS AS ERK INHIBITORS AND THEIR USE 2020
  • Li, Yi
  • Liu, Ning
  • Yu, Tao
  • Wu, Chengde
  • Li, Jian
  • Chen, Shuhui
RU2800042C1
BICYCLIC COMPOUND AS RIP-1 KINASE INHIBITOR AND ITS USE 2020
  • Wei, Wei
  • Li, Peng
  • He, Haiying
  • Chen, Shuhui
RU2800652C2
PDE4 INHIBITOR 2017
  • Luo, Yunfu
  • Yang, Chundao
  • Lei, Maoyi
  • Liu, Ling
  • Hu, Guoping
  • Li, Jian
  • Chen, Shuhui
RU2743126C2
TRICYCLIC COMPOUNDS AFFECTING CRBN PROTEINS 2019
  • Lej, Maoi
  • Lo, Yunfu
  • Syuj, Yuj
  • Chzhan, Goli
  • Yuj, Chzhitszyuan
  • Li, Tszyan
  • Chen, Shukhuej
RU2801068C2
THIOPHENE COMPOUND, ITS PRODUCTION METHOD AND ITS PHARMACEUTICAL APPLICATION 2017
  • Wang, Jianfei
  • Zhang, Yang
  • Zhu, Wenyuan
  • Chen, Shuhui
RU2709473C1
FGFR INHIBITOR AND ITS MEDICAL USE 2018
  • Wang, Yikai
  • Zhang, Yang
  • Chen, Zhengxia
  • Chen, Linlin
  • Feng, Tao
  • Huang, Rongxin
  • Li, Qiu
  • Li, Deyao
  • Sun, Jikui
  • Xu, Yangyang
  • Li, Jie
  • Li, Jian
  • Chen, Shuhui
RU2771311C2
PYRIDOPYRIMIDINE COMPOUNDS ACTING AS DOUBLE INHIBITORS OF mTORC 1/2 2018
  • Chen, Kevin X
  • Chen, Zhaoguo
  • Zhang, Li
  • Yu, Yanxin
  • Zhou, Kai
  • Hu, Boyu
  • Wang, Xiaofei
  • Hu, Guoping
  • Li, Jian
  • Chen, Shuhui
RU2771201C2
ALPHA-AMINOAMIDE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS THEREWITH 2015
  • Pak Ki Duk
  • Li Chkhanchon Dzhastin
  • Kim Ton Chin
  • Pe E Nim
  • Chkhu Khen A
  • Min Sun Chun
  • Kan En Ko
  • Kim Yun Ken
  • Sun Khe Chon
  • Chkhve Chi Von
  • Nam Min Kho
  • Kho Chon Yun
  • En Sol Ki
  • Chan Bo Ko
  • Chu Yn Chi
  • Cho Son Mi
  • Pak Chon-Khen
RU2673622C2
2,3-DIHYDRO-1H-PYRROLISINE-7-FORMAMIDE DERIVATIVE AND ITS APPLICATIONS 2019
  • Khe, Khajin
  • Sya, Tszyankhua
  • Gun, Chzhen
  • Li, Tszyan
  • Chen, Shukhuej
RU2792726C2
PYRIMIDINE DERIVATIVES AGAINST INFLUENZA VIRUS 2017
  • Syun, Tszian
  • Lun, Chaofen
  • Van, Tszintszin
  • Chen, Syaosin
  • Chen, Kevin Kh
  • Se, Chen
  • Li, Pen
  • Pen, Syuantszya
  • Li, Tszyan
  • Chen, Shukhuej
RU2727772C1

RU 2 805 569 C1

Authors

Li, Yi

Liu, Ning

Yu, Tao

Wu, Chengde

Li, Jian

Chen, Shuhui

Dates

2023-10-19Published

2020-12-07Filed