FIELD: organic chemistry.
SUBSTANCE: new biologically active compounds - substituted pyrido[b]pyrrolo[1,2-d][1,4]diazepines, namely 10-methyl-6,7-dihydro-5H-pyrido[2 ,3-b]pyrrolo[1,2-d][1,4]diazepine of Formula 1, which has antimycotic activity, which suggests its use in medicine as a drug with antimycotic properties. The use of 10-methyl-6,7-dihydro-5H-pyrido[2,3-b]pyrrolo[1,2-d][1,4]diazepine of Formula (1) as an antifungal agent against yeast fungi is presented.
EFFECT: invention provides 10-methyl-6,7-dihydro-5H-pyrido[2,3- b]pyrrolo[1,2-d][1,4]diazepine of Formula (1), which has a pronounced antimycotic effect and low toxicity.
1 cl, 1 tbl, 3 ex
| Title | Year | Author | Number |
|---|---|---|---|
| APPLICATION OF 5-[(1H-INDOL-3-YL)METHYL]-7-METHYL-2,3-DIHYDRO-1H-PYRROLO[1,2-D][1,4]DIAZEPIN-4(5H)-ONE AS AN ANTIFUNGAL AGENT FOR YEASTS | 2023 |
|
RU2803571C1 |
| USE OF 1-METHYL-4,5-DIHYDRO-6H-PYRIDO[1,2-a][1,4]BENZODIAZEPINE-6-ONE AS ANTIFUNGAL AGENT AGAINST YEASTS | 2023 |
|
RU2809026C1 |
| USE OF 7-METHYL-2-(4-METHYLPHENYL)-1,2,4,5-TETRAHYDRO-3H-PYRROLO[1,2-a][1,4]DIAZEPIN-3-ONE AS AN ANTIFUNGAL AGENT AGAINST YEAST FUNGI | 2023 |
|
RU2809053C1 |
| USE OF 5-(4-METOXYPHENYL)-7-METHYL-1,2,4,5-TETRAHYDRO-3H-PYRROLO[1,2-a][1,4]DIAZEPIN-3-ONE AS AN ANTIFUNGAL AGENT AGAINST YEAST FUNGI | 2023 |
|
RU2810715C1 |
| USE OF 1-METHYL-5-(4-CHLOROPHENYL)-4,5-DIHYDRO-6H-PYRROLO[1,2-a][1,4]BENZODIAZEPIN-6-ONE AS AN ANTIFUNGAL AGENT AGAINST YEAST FUNGI | 2023 |
|
RU2809148C1 |
| USE OF 7-METHYL-5-[4-(TRIFLUOROMETHYL)PHENYL]-1,2,4,5-TETRAHYDRO-3H-PYRROLO[1,2-a][1,4]DIAZEPIN-3-ONE AS AN ANTIFUNGAL AGENT AGAINST YEAST FUNGI | 2023 |
|
RU2808981C1 |
| USE OF 2-METHYL-4-[7-(TRIFLUOROMETHYL)PHENYL]-1,2,4,5-TETRAHYDRO-3H-PYRROLO[1,2-a][1,4]DIAZEPIN-3-ONE AS ANTIFUNGAL AGENT AGAINST YEAST FUNGI | 2023 |
|
RU2809051C1 |
| USE OF 1-METHYL-8,9-DIMETHOXY-4,5-DIHYDRO-6H-PYRROLO[1,2-A][1,4]BENZODIAZEPIN-6-ONE AS AN ANTIFUNGAL AGENT AGAINST YEAST FUNGI | 2023 |
|
RU2808993C1 |
| APPLICATION OF 5-ISOPROPYL-7-METHYL-2,3-DIHYDRO-1H-PYRROLO[1,2-d][1,4]DIAZEPIN-4(5H)-ONE AS ANTIBACTERIAL AGENT AGAINST GRAM-POSITIVE MICROORGANISMS | 2022 |
|
RU2784439C1 |
| USE OF 4,6-DIMETHYL-1,2-DIHYDROPYRROLO[1,2-a]PYRAZIN-3(4H)-ONE AS AN ANTIFUNGAL AGAINST YEASTS | 2023 |
|
RU2806191C1 |
