APPLICATION OF 10-METHYL-6,7-DIHYDRO-5H-PYRIDO[2,3-b]-PYRROLO[1,2-d][1,4]DIAZEPINE AS AN ANTIFUNGAL AGENT AGAINST YEASTS Russian patent published in 2023 - IPC A61K31/551 A61P31/10 

Abstract RU 2803600 C1

FIELD: organic chemistry.

SUBSTANCE: new biologically active compounds - substituted pyrido[b]pyrrolo[1,2-d][1,4]diazepines, namely 10-methyl-6,7-dihydro-5H-pyrido[2 ,3-b]pyrrolo[1,2-d][1,4]diazepine of Formula 1, which has antimycotic activity, which suggests its use in medicine as a drug with antimycotic properties. The use of 10-methyl-6,7-dihydro-5H-pyrido[2,3-b]pyrrolo[1,2-d][1,4]diazepine of Formula (1) as an antifungal agent against yeast fungi is presented.

EFFECT: invention provides 10-methyl-6,7-dihydro-5H-pyrido[2,3- b]pyrrolo[1,2-d][1,4]diazepine of Formula (1), which has a pronounced antimycotic effect and low toxicity.

1 cl, 1 tbl, 3 ex

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RU 2 803 600 C1

Authors

Uchuskin Maksim Grigorevich

Mendogralo Elena Iurevna

Makarov Anton Sergeevich

Nikiforova Elena Aleksandrovna

Rubtsov Aleksandr Evgenevich

Nesterova Larisa Iurevna

Tkachenko Aleksandr Georgievich

Ovchinnikova Olga Sergeevna

Dates

2023-09-18Published

2023-03-22Filed