USE OF 1-METHYL-5-(4-CHLOROPHENYL)-4,5-DIHYDRO-6H-PYRROLO[1,2-a][1,4]BENZODIAZEPIN-6-ONE AS AN ANTIFUNGAL AGENT AGAINST YEAST FUNGI Russian patent published in 2023 - IPC C07D487/04 A61K31/5517 A61P31/10 

Abstract RU 2809148 C1

FIELD: organic chemistry and pharmacology.

SUBSTANCE: invention relates to the use of substituted pyrrolo[1,2-a][1,4]benzodiazepines, which have antimycotic activity against yeast fungi. The use of 1-methyl-5-dihydro-6H-pyrrolo[4-a][4,5]benzodiazepin-1,2-one as an antifungal agent against yeast fungi is disclosed.

EFFECT: invention provides effective antimycotic activity against yeast fungi and has low toxicity.

1 cl, 1 tbl, 3 ex

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RU 2 809 148 C1

Authors

Uchuskin Maksim Grigorevich

Mendogralo Elena Iurevna

Nesterova Larisa Iurevna

Tkachenko Aleksandr Georgievich

Makarov Anton Sergeevich

Nikiforova Elena Aleksandrovna

Rubtsov Aleksandr Evgenevich

Sorotskaia Liudmila Nazarovna

Dates

2023-12-07Published

2023-04-27Filed