USE OF 1-METHYL-8,9-DIMETHOXY-4,5-DIHYDRO-6H-PYRROLO[1,2-A][1,4]BENZODIAZEPIN-6-ONE AS AN ANTIFUNGAL AGENT AGAINST YEAST FUNGI Russian patent published in 2023 - IPC C07D487/04 C07D243/14 A61K31/5517 A61P31/10 

Abstract RU 2808993 C1

FIELD: organic chemistry.

SUBSTANCE: use of 1-methyl-8,9-dimethoxy-4,5-dihydro-6H-pyrrolo[1,2-a][1,4]benzodiazepin-6-one of Formula 1:

as an antifungal agent against yeast fungi.

EFFECT: proposed use of 1-methyl-8,9-dimethoxy-4,5-dihydro-6H-pyrrolo[1,2-a][1,4]benzodiazepin-6-one, which has pronounced antimycotic activity against yeast fungi, as well as low toxicity.

1 cl, 3 ex, 1 tbl

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RU 2 808 993 C1

Authors

Uchuskin Maksim Grigorevich

Mendogralo Elena Iurevna

Nesterova Larisa Iurevna

Tkachenko Aleksandr Georgievich

Makarov Anton Sergeevich

Nikiforova Elena Aleksandrovna

Rubtsov Aleksandr Evgenevich

Sorotskaia Liudmila Nazarovna

Dates

2023-12-05Published

2023-04-26Filed