USE OF 4,6-DIMETHYL-1,2-DIHYDROPYRROLO[1,2-a]PYRAZIN-3(4H)-ONE AS AN ANTIFUNGAL AGAINST YEASTS Russian patent published in 2023 - IPC A61K31/498 C07D487/04 A61P31/10 

Abstract RU 2806191 C1

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to the use of 4,6-dimethyl-1,2-dihydropyrrolo[1,2-a]pyrazin-3(4H)-one of formula 1 as an antifungal agent against the yeast Candida albicans. Compound 1 has antimycotic activity, as well as low toxicity, which allows it to be used in medicine as a medicinal product with antimycotic properties.

EFFECT: use of 4,6-dimethyl-1,2-dihydropyrrolo[1,2-a]pyrazin-3(4h)-one as an antifungal against yeasts.

1 cl, 1 tbl, 3 ex

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RU 2 806 191 C1

Authors

Uchuskin Maksim Grigorevich

Sorotskaia Liudmila Nazarovna

Mendogralo Elena Iurevna

Makarov Anton Sergeevich

Nikiforova Elena Aleksandrovna

Rubtsov Aleksandr Evgenevich

Nesterova Larisa Iurevna

Tkachenko Aleksandr Georgievich

Batuev Roman Vladislavovich

Dates

2023-10-27Published

2023-03-22Filed