FIELD: pharmaceuticals.
SUBSTANCE: invention relates to a heteroaromatic amide derivative represented by the general formula (I-E2), pharmaceutical compositions, agents having inhibitory activity against Nav1.7, as well as the use of a heteroaromatic amide derivative or a pharmacologically acceptable salt thereof according to any one of claims 1–7 for the manufacture of a pharmaceutical composition having inhibitory activity against Nav1.7, used to prevent or eliminate the pain.
EFFECT: obtaining new compounds that have inhibitory activity against Nav1.7, which can be used to prevent or eliminate the pain.
17 cl, 99 tbl
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