USE OF MANNICH BASES BASED ON FUSIDIC ACID AS COMPOUNDS WITH ANTI-TUMOUR ACTIVITY Russian patent published in 2024 - IPC C07C215/50 A61K31/575 A61K31/58 A61P35/00 

Abstract RU 2819293 C1

FIELD: medicine.

SUBSTANCE: invention relates to medicine, and discloses the use of Mannich bases based on fusidic acid of formula (1) – (4) as compounds exhibiting high anti-tumour activity in vitro with respect to five human cancer cell lines HepG2, HCT-116, SH-SY5Y, MCF-7 and A549.

EFFECT: providing high anti-tumour activity in vitro with respect to five human cancer cell lines: HepG2, HCT-116, SH-SY5Y, MCF-7 and A549.

1 cl, 1 tbl, 2 ex

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RU 2 819 293 C1

Authors

Salimova Elena Viktorovna

Parfenova Liudmila Viacheslavovna

Ishmetova Diana Valievna

Zainullina Liana Fanzilevna

Vakhitova Iuliia Venerovna

Dates

2024-05-16Published

2023-06-22Filed