FIELD: chemistry.
SUBSTANCE: present invention relates to a compound of formula (Ia) or a pharmaceutically acceptable salt thereof
,
where in formula (Ia) R1 is phenyl, optionally substituted with a group selected from halogen, C1-6 alkyl and C1-6 alkyloxy; R2 is C1-3 alkyl, 5–6-membered heteroaryl containing 1 heteroatom selected from nitrogen, oxygen and sulphur, or phenyl, optionally substituted with a group selected from halogen, C1-6 alkyl and C1-6 alkyloxy; and Het is pyrazol-4-yl, as well as to a method of producing compounds of formula (Ia) and to a pharmaceutical composition containing a compound of formula (Ia).
EFFECT: there are prepared new compounds which can be used for treating cancer, such as human glioblastoma, human breast duct carcinoma, human liver and embryonic kidney carcinoma.
6 cl, 2 tbl, 4 ex
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