HETEROCYCLIC AMIDE COMPOUND, PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, METHOD FOR PREPARATION AND USE THEREOF Russian patent published in 2024 - IPC C07D491/48 A61K31/4188 A61P35/00 A61P31/00 

Abstract RU 2823875 C1

FIELD: chemistry.

SUBSTANCE: invention relates to a heterocyclic amide compound of general formula I, where A, B, C, R1-R4, R2’-R4’, RB are defined in the claims, and a pharmaceutically acceptable salt thereof, to a method for production thereof.

EFFECT: invention discloses use of the compound for preparing a preparation for treating diseases associated with STING activity, for preparing an immunological adjuvant and for preparing a preparation for activating STING.

16 cl, 2 dwg, 2 tbl, 26 ex

Formula I

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RU 2 823 875 C1

Authors

Duan, Wenhu

Geng, Meiyu

Zhang, Huibin

Xie, Zuoquan

Zhou, Jinpei

Yang, Yifei

Wang, Xiyuan

Yang, Xiaojun

Zhang, Yan

Hu, Zhaoxue

Ding, Jian

Dates

2024-07-30Published

2020-09-21Filed