POLYPEPTIDE HAVING MMR-2 INHIBITORY ACTION Russian patent published in 2024 - IPC C07K7/06 A61K38/07 A61K38/08 A61P35/00 C12N9/99 

Abstract RU 2828218 C1

FIELD: chemistry.

SUBSTANCE: invention relates to a substituted polypeptide of formula I'-B, where AA1-AA5, WC, RC are defined in the claims, or a pharmaceutically acceptable salt thereof, which has the inhibitory effect of MMP2. Also disclosed is a pharmaceutical preparation, an MMP2 inhibitor and a drug having MMP2 inhibitory activity.

EFFECT: disclosed is a polypeptide having mmr-2 inhibitory action.

5 cl, 53 tbl, 9 ex

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RU 2 828 218 C1

Authors

Khayasi, Masato

Takeuti, Tomoki

Nomura, Yusaku

Tamita, Tomoko

Simono, Rie

Dates

2024-10-08Published

2020-11-06Filed