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2 841 063

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IPC

C07D405/14(2006-01-01)

A61K31/37(2006-01-01)

A61P31/16(2006-01-01)

(21) (22)

Application

2024117574, 2024-06-26

(24)

Start date

2024-06-26

(22)

Actual filing date

2024-06-26

(45)

Published

2025-06-02

(72)

Inventor

Shults Elvira EduardovnaShtro Anna AndreevnaGarshinina Anzhelika ValerevnaSavelev Viktor AleksandrovichGalochkina Anastasiia Valerevna

(73)

Holder

Federalnoe Gosudarstvennoe Biudzhetnoe Uchrezhdenie Nauki Novosibirskii Institut Organicheskoi Khimii Im. N.N. Vorozhtsova Sibirskogo Otdeleniia Rossiiskoi Akademii Nauk So Ran)Federalnoe Gosudarstvennoe Biudzhetnoe Uchrezhdenie Institut Grippa Imeni A.A. Smorodintseva» Ministerstva Zdravookhraneniia Rossiiskoi Federatsii

2-(1,2,3-TRIAZOLYL)SUBSTITUTED LINEAR FUROCOUMARINS HAVING ANTIVIRAL ACTIVITY AGAINST INFLUENZA A/H1N1 VIRUS Russian patent published in 2025 - IPC C07D405/14 A61K31/37 A61P31/16

Abstract RU 2841063 C1

FIELD: chemistry.

SUBSTANCE: invention relates to use of 2-(1,2,3-triazol-1-yl)substituted derivatives of linear oreozelon furocoumarin of general formula (I), wherein the compound of formula (I) is Ia, where R¹ is a fragment specified in the claims, and R² is H; and Ib, where R¹ is a fragment (a) and R² is a fragment of (b) as an agent having inhibitory activity on influenza A/H1N1 virus.

EFFECT: more effective suppression of influenza virus reproduction and wider range of influenza virus reproduction inhibitors for overcoming drug resistance of current viral strains.

1 cl, 1 dwg, 1 tbl, 4 ex

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RU 2 841 063 C1

Authors

Shults Elvira Eduardovna

Shtro Anna Andreevna

Garshinina Anzhelika Valerevna

Savelev Viktor Aleksandrovich

Galochkina Anastasiia Valerevna

Dates

2025-06-02—Published

2024-06-26—Filed