FIELD: organic chemistry. SUBSTANCE: product: 3-(1,2-benzisoxazole-3-yl)-4-pyridamines of the general formula I (R1), where R2 and - hydrogen or lower alkyl. Compounds of the general formula I are synthesized by cyclization of corresponding substituted o-halogenphenylmethaneoxime in the presence of base in the medium of lower alcohol. Synthesized compounds are used in medicine. EFFECT: improved method of synthesis of compounds indicated above. 3 tbl
Title |
Year |
Author |
Number |
BENZISOTHIAZOLE- OR BENZISOXAZOLE-3-CARBOXAMIDES OR THEIR PHARMACEUTICALLY ACCEPTABLE SALTS, METHODS OF THEIR SYNTHESIS AND PHARMACEUTICAL COMPOSITION SHOWING ANTIPSYCHOTIC ACTIVITY |
1992 |
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- Dzhon G.Dzhurkak[Us]
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TETRAHYDROACRIDINE DERIVATIVES, PROCESSES FOR PREPARATION THEREOF (VARIANTS), TETRAHYDROACRIDINONE DERIVATIVES, DIHYDROBENZOXAROLE DERIVATIVE AND PHARMACEUTIC COMPOSITION HAVING EFFECT OF EASING OR ELIMINATING MEMORY DYSFUNCTION |
1992 |
- Gregori Majkl Shatski[Us]
- Kevin Dzhejms Kaples[Us]
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1992 |
- Richard Charl'Z Ehffland[Us]
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PROCESS FOR PREPARING ISOMERS, OR PHARMACEUTICALLY ACCEPTABLE SALTS, AND ALDEHYDE AS AN INTERMEDIATE PRODUCT IN THE 1-ALKYL, 1-ALKENYL OR 1-ALKYNYLARYL-2-AMINO-1, 3- PROPANEDIOL SYSTEM |
1991 |
- Dzhon Dzhozef Tidzheler[Us]
- Barbara Sivi Rokman[Us]
- Rassell Richard Li Khejmer[Us]
- Brajan Skott Frid[Us]
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RU2024493C1 |
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1990 |
- Dzhozef Tomas Strupchevski[Us]
- Grover Kleveland Khelslej[Us]
- Julin Chiang[Us]
- Kennet Dzh.Bordeo[Us]
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RU2062776C1 |
DERIVATIVES OF N-(ARYLOXYALKYL)-HETEROARYLPIPERIDINE AND HETEROARYLPIPERAZINE AND PHARMACEUTICAL COMPOSITION BASED ON THEREOF |
1990 |
- Dzhozef Tomas Strupchevski
- Grover Kleveland Khelslej
- Julin Chiang
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1-ALKYL, 1-ALKENYL OR 1-ALKYNYLARYL-2-AMINO-1,3-PROPANEDIOLS OR THEIR OPTICAL ISOMERS OR PHARMACEUTICALLY ACCEPTABLE SALTS AND METHOD OF THEIR SYNTHESIS |
1992 |
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1992 |
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METHOD OF SYNTHESIS OF AMINOCARBONYLCARBAMATES |
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