3-(1,2-BENZISOXAZOLE-3-YL)-4-PYRIDAMINES SHOWING ANALGETIC, ANTICHOLINE ESTERASE AND DERMATOLOGICAL ACTIVITIES Russian patent published in 1994 - IPC

Abstract RU 2012561 C1

FIELD: organic chemistry. SUBSTANCE: product: 3-(1,2-benzisoxazole-3-yl)-4-pyridamines of the general formula I (R1), where R2 and - hydrogen or lower alkyl. Compounds of the general formula I are synthesized by cyclization of corresponding substituted o-halogenphenylmethaneoxime in the presence of base in the medium of lower alcohol. Synthesized compounds are used in medicine. EFFECT: improved method of synthesis of compounds indicated above. 3 tbl

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RU 2 012 561 C1

Authors

Dzhozef Tomas Klajn[Us]

Richard Charl'Z Ehffland[Us]

Dates

1994-05-15Published

1991-08-12Filed