FIELD: organic chemistry. SUBSTANCE: product: heterocyclic compound of the formula (I) where R1 and R2 - hydrogen; R3 - hydrogen, hydroxyl, methoxyl, C1-C3-alkyl or the group XR4 at X - oxygen or S(O)n; n = 0 or 1; R4-C1-C3-alkyl, cyclopentyl or phenyl, or if X - oxygen then R4 can mean AlkNR5R6 where Alk - C2-alkylene chain; R5 and R6 are independent - hydrogen or R5 - iminomethyl and R6 - hydrogen or R3 - the group (CH)(CH)mNR7R8 at m= 0 or 1, and R7 and R8 are independent - hydrogen or C1-C4--alkyl, or R7 - acetyl or iminomethyl, and R8 - hydrogen, or R3 - carbon atom to which it is connected and represents keto-group or its ketal-derivative, and also their physiologically acceptable salts involving internal salt if it is possible, and metabolically labile esters. Synthesized compounds were used in medicine and veterinary. EFFECT: improved method of synthesis. 6 cl, 4 tbl
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Authors
Dates
1996-02-10—Published
1992-06-04—Filed