METHOD OF ENANTIOSELECTIVE SYNTHESIS OF PHENYLISOSERINE DERIVATIVES Russian patent published in 1997 - IPC

Abstract RU 2086538 C1

FIELD: organic chemistry. SUBSTANCE: invention relates to method of enantioselective synthesis of phenylisoserine derivatives of the general formula (I) where: R means phenyl or tert.-butoxy; R′ means protective group for alcoholic function. Compounds of the general formula (I) can be used for synthesis of taxane derivatives that show antitumor and antileukemic activity. EFFECT: improved method of synthesis.

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RU 2 086 538 C1

Authors

Arlen Korrea[Br]

Zhan-Noel' Deni[Be]

Ehndrju-Ehlliot Grin[Us]

Dehvid Skott Grirson[Ca]

Dates

1997-08-10Published

1991-05-21Filed