CYCLIC UREAS, METHOD OF INHIBITION OF RETROVIRUS GROWTH AND PHARMACEUTICAL COMPOSITION Russian patent published in 1999 - IPC

Abstract RU 2131420 C1

FIELD: organic chemistry, pharmacy. SUBSTANCE: invention describes new cyclic derivatives of urea of the general formula (I) where values W, R4,R,R5,R6,R7,R and n are given in p. 1 of the invention claims. Synthesized compounds can be used as inhibitors of retroviral protease activity. Invention describes a pharmaceutical composition based on compounds of the formula (I) and a method of inhibition of retrovirus growth using compounds of the formula (I). EFFECT: enhanced inhibitory activity of compounds. 20 cl, 2 tbl, 22 ex

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Authors

Patrik Juk-Sun Lehm

Charl'Z Dzhozef Ajrmehnn

Karl Nikolas Khodzh

Prabkhakar Kondadzhi Dzhadkhav

Dzhordzh Vinsent Delukka

Dates

1999-06-10Published

1992-10-13Filed