N,N′-SUBSTITUTED IMIDOCARBONIMIDE DIAMIDES, PROPHYLACTIC COMPOSITION, COMPOSITION FOR DECREASE OF INFECTION LEVEL Russian patent published in 1999 - IPC

Abstract RU 2133737 C1

FIELD: organic chemistry, pharmacy. SUBSTANCE: invention describes the novel N,N′-substituted imidocarbonimide diamides of the general formula (I) where R1 means bivalent nonsubstituted lower aliphatic group; R3 means C1-C10-alkyl that is substituted with lower alkyl of phenyl that is substituted with halogen atom; R5 means phenyl or benzyl that can be mono- or poly-substituted with halogen atom, nitro-group, lower alkyl, lower alkoxy-group or naphthyl; R6 means hydrogen atom; R7 means hydrogen atom, C1-C10-alkyl, alkanoyl; Y means oxygen or sulfur atom; q = 1; m = 1, their pharmaceutically acceptable additive salts or hydrates of indicated salts. The above indicated compounds show antiparasitic and antibacterial activity. Invention describes the prophylactic composition based on compounds of the formula (I) for decrease of infection level in patients. EFFECT: enhanced effectiveness of compounds and composition. 21 cl, 7 tbl, 8 ex

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RU 2 133 737 C1

Authors

Krejg Kehnfild

Dehvid P.Dzhakobus

Nejl Dzh. Levis

Dates

1999-07-27Published

1993-01-19Filed