FIELD: medicine, pharmaceutics.
SUBSTANCE: present invention refers to medicine and described a water-based liquid composition for activation of intraocular penetration of a compound of formula (I) containing an amide compound, and an agent forming an ionic pair. What is also described is a method for activation of intraocular penetration of the compound presented by formula (I), and using the compound prepared by formula (I).
EFFECT: invention provides activation of penetration of the compound of formula (I), as well as maintaining the pre-set concentration of the drug preparation, even if a periodicity of the composition administration is reduced.
14 cl, 7 tbl, 2 dwg, 4 ex
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