FIELD: organic chemistry, pharmacy. SUBSTANCE: invention relates to derivatives of N-phenyl-2-pyrimidineamine of the formula (I) 
where R0 - hydrogen, halogen atom, lower alkoxy-group or lower alkyl; R1 means N-aminoalkylcarbamoyl, N-hydroxyalkylcarbamoyl, hydrazino-, cyclohexylamino-group possibly substituted with amino-, piperazinyl-, morpholinyl- or alkylamino-group that inhibit protein kinase activity at high selectivity degree. EFFECT: improved method of synthesis, high selective inhibition. 15 cl, 1 tbl, 29 ex
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