FIELD: organic chemistry, pharmacy. SUBSTANCE: invention relates to derivative of benzimidazole of the formula (I) where R3 - a residue of the formula (a) where R11 - pyridyl, imidazole, furanyl, pyrimidinyl, thienyl or thiazolyl possibly substituted with amino-group; one of R6 or R7 - hydrogen atom and another means -CR'=NOR'' where each of R' and R'' - hydrogen atoms, alkyl, alkenyl or alkynyl, or its pharmaceutically acceptable salt or oxide or a pharmaceutical composition based on said that provides modulation of GAOA-receptor complex of the central nervous system of living organism. EFFECT: effective modulation of receptor complex. 8 cl, 1 tbl, 5 dwg, 34 ex
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