CARBOHYDRATE DERIVATIVES, PHARMACEUTICAL COMPOSITION BASED ON THEREOF Russian patent published in 2002 - IPC

Abstract RU 2183638 C2

FIELD: organic chemistry, carbohydrates, pharmacy. SUBSTANCE: invention relates to a carbohydrate derivative of the general formula (I) where R means H or CH2OSO-3

; R2 and R3 mean independently H, (1-6C)-alkyl or SO-3
; R4 means OSO-3
; n = 0 or 1; p = 1 or 2, or to its a pharmaceutically acceptable salt. Compounds show antithrombosis activity. Also, invention proposes a pharmaceutical composition comprising indicated carbohydrate derivative used for treatment and prophylaxis or diseases mediated or associated with thrombin. EFFECT: valuable medicinal properties of carbohydrate derivatives. 8 cl

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RU 2 183 638 C2

Authors

Van Bukkel Konstant Adrian Anton

Vesterdejn Piter

Dates

2002-06-20Published

1997-05-07Filed