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Application

2002128954/15, 2002-10-29

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Start date

2002-10-29

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Actual filing date

2002-10-29

(45)

Published

2004-02-10

(72)

Inventor

Sernov L.N.Skachilova S.Ja.Blinov D.S.Druzhinina V.V.Kostin Ja.V.Shilova E.V.

(73)

Holder

Gosudarstvennoe Unitarnoe Predprijatie Nauchnyj Tsentr Po Bezopasnosti Biologicheski Aktivnykh Veshchestv"

DERIVATIVES OF 2-DIETHYLAMINO-2,6-DIMETHYLPHENYLACETAMIDE ELICITING ANTI-ARRHYTHMIC ACTIVITY Russian patent published in 2004 - IPC

Abstract RU 2223263 C1

FIELD: organic chemistry, medicine, cardiology, pharmacy. SUBSTANCE: invention proposes new derivatives of 2-diethylamino- -2¹,6¹-dimethylphenylacetamide with anti-arrhythmic activity. New derivatives represent new lidocaine salts: L-arginate, L-glutaminate, N-acetyl-L-glutaminate, 2- aminopropionate, aminoacetate, succinate, N-acetylcysteinate and β--phenyl--α--aminopropionate with enhanced effectiveness and safety as compared with lidocaine hydrochloride. EFFECT: expanded assortment of agents with indicated designation, valuable medicinal properties of derivatives. 4 tbl, 9 ex

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RU 2 223 263 C1

Authors

Sernov L.N.

Skachilova S.Ja.

Blinov D.S.

Druzhinina V.V.

Kostin Ja.V.

Shilova E.V.

Dates

2004-02-10—Published

2002-10-29—Filed