FIELD: organic chemistry, medicine.
SUBSTANCE: invention describes derivatives of 1,2,4,5-tetrahydrobenzo[d]azepines of the general formula (I):
wherein X means -N=, =N-, -N<, >C= or =C<; Y means -N=, =N-, -NH-, -CH= or =CH-; dotted line can mean a bond; radicals R1-R16 are described in the invention claim, and also their pharmaceutically acceptable salts in their racemic and optically active form. Also, invention describes a medicinal agent that can be used in treatment or prophylaxis of acute and/or chronic neurological disorders. Invention provides preparing new compounds eliciting useful biological properties.
EFFECT: valuable medicinal properties of compounds.
13 cl, 1 tbl, 276 ex
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Authors
Dates
2004-11-20—Published
2000-08-04—Filed