FIELD: organic chemistry, chemical technology.
SUBSTANCE: invention describes a method for preparing 1,3-oxathiolan nucleosides or a method for preparing derivatives of 1,3-oxathiolanyl-5-one that involve effective methods for formation of 1,3-oxathiolan ring followed by condensation of 1,3-oxathiolan with pyrimidine or purine base. Using indicated methods these compounds can be synthesized as separate enantiomers with high selectivity.
EFFECT: improved preparing methods.
27 cl, 3 dwg, 16 ex
Title |
Year |
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Number |
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