METHOD FOR PREPARING 1,3-OXATHIOLAN NUCLEOSIDE, METHOD FOR PREPARING DERIVATIVE OF 1,3-OXATHIOLANYL-5-ONE Russian patent published in 2005 - IPC

Abstract RU 2244712 C2

FIELD: organic chemistry, chemical technology.

SUBSTANCE: invention describes a method for preparing 1,3-oxathiolan nucleosides or a method for preparing derivatives of 1,3-oxathiolanyl-5-one that involve effective methods for formation of 1,3-oxathiolan ring followed by condensation of 1,3-oxathiolan with pyrimidine or purine base. Using indicated methods these compounds can be synthesized as separate enantiomers with high selectivity.

EFFECT: improved preparing methods.

27 cl, 3 dwg, 16 ex

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RU 2 244 712 C2

Authors

Pehjnter Dzhordzh R.

Liotta Dennis K.

Ehlmond Merrik

Kliri Dehrril

Sorija Khose

Shnajdman Markos Luis

Dates

2005-01-20Published

1999-08-12Filed