DERIVATIVES OF INDOLYL-3-GLYOXYLIC ACID - COMPOUNDS ELICITING ANTITUMOR ACTIVITY, PHARMACEUTICAL COMPOSITION, ANTITUMOR AGENT (VARIANTS) Russian patent published in 2005 - IPC

Abstract RU 2262339 C2

FIELD: organic chemistry, medicine, oncology, pharmacy.

SUBSTANCE: invention relates to applying N-substituted indole-3-glyoxylamides as antitumor agents. For administration invention proposes the following medicinal formulations: tablet, lozenges, capsule, solution for infusion or ampoule, suppository, plaster, composition for inhalation, suspension, cream and ointment. Compounds can be used in form of physiologically active acid-additive salts or N-oxides. Invention provides expanding assortment of antitumor medicinal agents.

EFFECT: valuable medicinal properties of compounds.

10 cl, 3 dwg, 6 tbl, 25 ex

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RU 2 262 339 C2

Authors

Bruneh Kaj

Gjunter Ehkkhard

Zelenyj Ishtvan

Nikel' Bernd

Rajkhert Ditmar

Shmidt Jurgen

Ehmig Peter

Dates

2005-10-20Published

1999-03-22Filed