FIELD: organic chemistry, medicine, pharmacy.
SUBSTANCE: invention relates to a conjugate target - compound chosen from the following group: and wherein means a target; each among R and R' means independently unsubstituted (C1-C20)-aliphatic group, substituted (C1-C20)-aliphatic group, unsubstituted aryl or substituted aryl wherein aryl is a radical chosen from the group comprising phenyl, naphthyl, tetrahydronaphthyl, indanyl, indenyl, pyridyl, pyrazinyl, pyrimidinyl, pyrrolyl, pyrazolyl, imidazolyl, thiazolyl, oxazolyl, isooxazolyl, thiadiazolyl, oxadiazolyl, thiophenyl, furanyl, quinolinyl, isoquinolinyl; m = 0, 1 or 2; n = 1 or 2. Also, invention describes library of compounds, method for identifying compounds, method for identifying the potential ligand. Proposed invention can promote to discovery of medicinal preparations.
EFFECT: valuable method for finding ligands.
20 cl, 8 dwg, 4 tbl, 21 ex
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Authors
Dates
2007-03-20—Published
2002-04-24—Filed