DEUTERATED 3-PIPERIDINOETHYLPHENYLKETONES, PHARMACEUTICAL COMPOSITION BASED ON THEREOF AND USING Russian patent published in 2007 - IPC C07D295/10 C07B59/00 A61K31/4453 A61P21/00 

Abstract RU 2296755 C2

FIELD: organic chemistry, medicine, pharmacy.

SUBSTANCE: invention relates to 3-piperidinoethylphenylketones of the general formula (I): wherein R means nondeuterated, mono- or multi-deuterated or perdeuterated alkyl comprising up to 3 carbon atoms; all radicals R' represent hydrogen atom, or all represent deuterium; radicals R'' represent independently of one another deuterium or hydrogen atom wherein at least one of radicals R, R' or R'' represents deuterium or comprises deuterium, and to their physiologically tolerant salts. Compounds of the formula (I) and their salts can be used in treatment of diseases associated with symptoms in muscular region, such as morbid reflex-muscular tensions of skeletal musculature and/or nervous-muscular convulsions.

EFFECT: valuable medicinal properties of compounds and pharmaceutical composition.

5 cl, 5 dwg, 10 ex

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RU 2 296 755 C2

Authors

Alken Rudol'F-Gizbert

Shtabingiz Tomas

Dates

2007-04-10Published

2002-04-29Filed