PAROXETINE DERIVATIVE Russian patent published in 2017 - IPC C07D405/12 A61K31/4525 A61P15/00 A61P25/24

Abstract RU 2616610 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a new compound represented by the formula (1)

wherein R¹ represents a hydrogen atom, or its pharmacologically acceptable salt which has improved inhibitory effect towards CYP, as well invention relates to a pharmaceutical composition based on this compound having the action of the selective inhibitor of serotonin reuptake , an antidepressant, and an agent for the treatment or prevention of premature ejaculation.

EFFECT: document describes a paroxetine derivative.

18 cl, 1 dwg, 4 tbl, 1 ex

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RU 2 616 610 C2

Authors

Tanaka Kejgo

Nisioka Tomoki

Dates

2017-04-18—Published

2013-01-29—Filed