ANTIMICROBIAL PRESERVATIVES FOR OBTAINING MULTIDOZE COMPOUNDINGS USING β-CYCLODEXTRINES FOR LIQUID MEDICINAL FORMS Russian patent published in 2008 - IPC A61K31/46 A61K47/10 A61K47/32 

Abstract RU 2332997 C2

FIELD: medicine; pharmacology.

SUBSTANCE: invention refers to pharmaceutical composition for treatment of disease, condition or disturbance requiring application of the antagonist of the neurokinin receptor containing therapeutically effective quantity of compound of the formula I or its pharmaceutically acceptable salt where the composition contains sulphopropyl ether of β-cyclodextrin, meta-cresol preservative and pharmaceutically acceptable medium. Also, the invention refers to application of the said composition and a method for treatment way of diseases requiring application of the antagonist of the neurokinin receptor.

EFFECT: maintenance of stability of a compounding and acceptable tolerance in the place of the product injection when using preservative for prevention of bacteriemic and fungoid growth in a compounding.

11 cl, 4 dwg, 9 tbl, 4 ex

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RU 2 332 997 C2

Authors

Adami Rodzher Kristofer

David Frederik

Vud Dzhulija Ehnn

Dates

2008-09-10Published

2005-01-17Filed