SOLID DOSAGE FORM OF CLOPIDOGREL AND METHOD FOR PREPARING THEREOF Russian patent published in 2010 - IPC A61K31/4365 A61K9/22 A61P7/02 

Abstract RU 2393862 C1

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to pharmaceutical industry and concerns a solid dosage form that exhibits the antiaggregatory activity and contains, wt %: clopidogrel hydrosulfate - 15-45; microcrystalline cellulose - 7-20; talc-1-3; sodium croscarmellose - 1-4; low-molecular polyvinylpyrrolidone - 0.3-10; stearic acid and/or its salts - 0.5-1; lactose - the rest, and a coating that contains, wt %: titanium dioxide - 8-30; polyethylene glycol - 6-28; talc - 5-25; carmine - 0.3-2.5; yellow aluminium lake - 0.05-1; red aluminium lake - 0.01-0.5; quinoline yellow aluminium lake - 0.01-0.05; polyvinyl alcohol - the rest. There is also disclosed a method for preparing the presented solid dosage form.

EFFECT: preparation of the solid dosage form that exhibits the antiaggregatory activity.

7 cl, 2 tbl

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Authors

Dates

2010-07-10Published

2009-03-05Filed