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(19)

(11)

2 403 245

(13)

(51)

IPC

C07D239/50(2006-01-01)

A61K31/505(2006-01-01)

A61P31/18(2006-01-01)

(21) (22)

Application

2007132179/04, 2006-01-27

(24)

Start date

2006-01-27

(22)

Actual filing date

2006-01-27

(45)

Published

2010-11-10

(72)

Inventor

Zhanssen Pol' Adrian JanKheres JanLevi Paulus JoannesLemans Rudol'FMuns Luk Jozef Rafaehl'

(73)

Holder

Tibotek Farmas'Jutikalz Ltd.

HIV INHIBITING DERIVATIVES OF 2-(4-CYANOPHENYLAMINO) PYRIMIDINE Russian patent published in 2010 - IPC C07D239/50 A61K31/505 A61P31/18

Abstract RU 2403245 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention relates to novel compounds, which have anti HIV-1 activity, of general formula (I) , where X stands for NH, as well as their pharmaceutically acceptable additive salt. Invention also relates to pharmaceutical composition, method of obtaining pharmaceutical composition and method of obtaining compound.

EFFECT: novel compounds possessing anti-HIV-1 activity.

5 cl, 7 dwg, 1 tbl, 14 ex

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RU 2 403 245 C2

Authors

Zhanssen Pol' Adrian Jan

Kheres Jan

Levi Paulus Joannes

Lemans Rudol'F

Muns Luk Jozef Rafaehl'

Dates

2010-11-10—Published

2006-01-27—Filed