HIV-INHIBITING 2-(4-CYANOPHENYL)-6-HYDROXYLAMINO-PYRIMIDINES Russian patent published in 2010 - IPC C07D239/48 C07D405/12 A61K31/505 A61P31/18 

Abstract RU 2401261 C2

FIELD: chemistry.

SUBSTANCE: invention relates to novel compounds of formula (I) and their pharmaceutically acceptable addition salts having HIV replication inhibiting properties. In formula (I), R1 is halogen; R2 and R3 each independently denotes C1-6-alkyl. The invention also relates to a method for synthesis of said compounds and a pharmaceutical composition.

EFFECT: increased effectiveness of derivatives.

7 cl, 6 ex

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RU 2 401 261 C2

Authors

De Kok Kherman Augustinus

Vigerink Pit Tom Bert Pol'

Dates

2010-10-10Published

2006-03-02Filed