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RU

(11)

2 416 599

(13)

C2

(51)

IPC

C07D207/32(2006-01-01)

C07C239/14(2006-01-01)

C07D213/56(2006-01-01)

C07D307/46(2006-01-01)

C07D333/22(2006-01-01)

C07D409/06(2006-01-01)

A61K31/34(2006-01-01)

A61K31/40(2006-01-01)

A61K31/5375(2006-01-01)

C07D213/50(2006-01-01)

C07D295/10(2006-01-01)

C07D307/80(2006-01-01)

C07D333/56(2006-01-01)

A61K31/16(2006-01-01)

A61K31/381(2006-01-01)

A61K31/44(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2007116098/04, 2005-09-30

(24)

Start date

2005-09-30

(22)

Actual filing date

2005-09-30

(45)

Published

2011-04-20

(72)

Inventor

Minuchchi SaverioPelichchi P'Er DzhuzeppeMaj AntonelloBallarini MarkoGarg'Julo GaehtanoMassa Sil'Vio

(73)

Holder

Dak S.R.L.

NOVEL HISTONE DEACETYLASE INHIBITORS Russian patent published in 2011 - IPC C07D207/32 C07C239/14 C07D213/56 C07D307/46 C07D333/22 C07D409/06 A61K31/34 A61K31/40 A61K31/5375 C07D213/50 C07D295/10 C07D307/80 C07D333/56 A61K31/16 A61K31/381 A61K31/44 A61P35/00 

Abstract RU 2416599 C2

FIELD: chemistry.

SUBSTANCE: present invention describes novel compounds of formula (I), where substitutes R1, R2, R3, Ar and A are described in the formula of invention, having histone deacetylase inhibiting activity, use thereof and methods for synthesis of said compounds.

EFFECT: improved composition properties.

15 cl, 72 ex, 9 tbl, 6 dwg

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RU 2 416 599 C2

Authors

Minuchchi Saverio

Pelichchi P'Er Dzhuzeppe

Maj Antonello

Ballarini Marko

Garg'Julo Gaehtano

Massa Sil'Vio

Dates

2011-04-20—Published

2005-09-30—Filed

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